Methoxy-PEPy

Description:
Methoxy-PEPy is a unique compound that acts as an allosteric ligand for kappa-opioid receptors. It is synthesized using a specific chemical synthesis method, making it a valuable research chemical. Methoxy-PEPy functions as a substrate inhibitor, blocking the activity of these receptors and preventing the binding of opioid peptides. This compound has been shown to be a noncompetitive antagonist for kappa-opioid receptors, inhibiting their function and reducing their binding affinity. Additionally, Methoxy-PEPy has demonstrated pharmacologic effects on glutamate release and electrophoresis in various studies. Its interaction with asparagine-linked oligosaccharides suggests potential therapeutic applications in modulating opioid receptor signaling pathways. Researchers interested in receptor binding and studying the effects of opioids will find Methoxy-PEPy to be an invaluable tool in their investigations.