Product Name :
GS 9973

Synonym :
6-(1H-Indazol-6-yl)-N-(4-morpholinophenyl)imidazo[1,2-a]pyrazin-8-amine

Chemical Name :

CAS NO.:
1229208-44-9

Molecular formula :
C23H21N7O

Molecular Weight:
411.47 g/mol

Classification :
MedChemExpress Products > Life Sciences > GS 9973

Description:
GS 9973 is a research drug that inhibits the activity of protein kinases, which are enzymes that regulate the function of other proteins. GS 9973 inhibits the activity of mcl-1, an effector protein in the apoptosis pathway and is currently being tested for its ability to inhibit cancer cells from spreading. GS 9973 has been shown to have a low risk of toxicity in humans and has been found to be safe for use in clinical trials with human pharmacokinetics. This drug also inhibits P-gp substrates, which prevents it from entering into the retina. The only side effects observed so far are eye disorders such as conjunctivitis and iritis.

Purity :
>98%

Specifications :
10 mM * 1 mL

Price.:
101

Price unit :
$

Inventory :
In stock

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